Kinase Inhibitors : Methods and Protocols - Kuster, Bernhard; SpringerLink (Online service) (Totowa, NJ : Humana Press : Imprint: Humana, 2012)
Targeting Cancer with Small Molecular Weight Kinase Inhibitors -- Small Molecule Protein and Lipid Kinase Inhibitors in Inflammation and Specific Models for their Evaluation -- Measuring the Activity of Leucine Rich Repeat Kinase 2 (LRRK2) - A Kinase Involved in Parkinson's Disease -- Measuring PI3K Lipid Kinase Activity -- A Fluorescence Polarization Assay for the Discovery of Inhibitors of the Polo-box Domain of Polo-like Kinase 1 -- Assessment of Hepatotoxicity Potential of Drug Candidate Molecules Including Kinase Inhibitors by Hepatocyte Imaging Assay Technology and Bile Flux Imaging Assay Technology -- Kinase Inhibitor Selectivity Profiling using Differential Scanning Fluorimetry -- Chemoproteomic Characterization of Protein Kinase Inhibitors using Immobilized ATP -- Proteome-wide identification of staurosporine-binding kinases using Capture Compound Mass Spectrometry -- Affinity Purification of Proteins Binding to Kinase Inhibitors Immobilised on Self Assembling Monolayers -- Kinase Inhibitor Profiling using Chemoproteomics -- Covalent Crosslinking of Kinases with Their Corresponding Peptide Substrates -- Receptor Tyrosine Kinase Inhibitor Profiling using Bead-based Multiplex Sandwich Immunoassays -- Monitoring Phosphoproteomic Response To Targeted Kinase Inhibitors Using Reverse-Phase Protein Microarrays -- Measuring Phosphorylation Specific Changes in Response to Kinase Inhibitors in Mammalian Cells Using Quantitative Proteomics -- Investigation of Acquired Resistance to EGFR-Targeted Therapies in Lung Cancer Using cDNA Microarrays.
Keywords: Pharmacology; Pharmacology/Toxicology.