Peptidomimetics Protocols - Kazmierski, Wieslaw M.; SpringerLink (Online service) (Totowa, NJ : Humana Press : Imprint: Humana, 1999)
Synthesis and Use of Pseudopeptides Derived from 1,2,4-Oxadiazole-, 1,3,4-Oxadiazole-, and 1,2,4-Triazole-based Dipeptidomimetics -- Synthesis of Aminobenzoic Acid-Based Nonpeptide Templates: Applications in Peptidomimetic Drug Discovery -- Synthesis of an Esterase-Sensitive Cyclic Prodrug of a Model Hexapeptide Having Enhanced Membrane Permeability and Enzymatic Stability Using an Acyloxyalkoxy Promoiety -- Synthesis of an Esterase-Sensitive Cyclic Prodrug of a Model Hexapeptide Having Enhanced Membrane Permeability and Enzymatic Stability Using a 3-(2?-Hydroxy-4?,6?-Dimethylphenyl)-3,3-Dimethyl Propionic Acid Promoiety -- Synthesis of Coumarin-Based, Esterase-Sensitive Cyclic Prodrugs of Opioid Peptides with Enhanced Membrane Permeability and Enzymatic Stability -- Azatides as Peptidomimetics: Solution and Liquid Phase Syntheses -- Synthesis of Cbz-Protected Ketomethylene Dipeptide Isosteres -- (E)-Alkene Peptide Bond Isosteres by Cuprate Opening of Vinyl Aziridines -- Syntheses of Norstatine, Its Analogs, and Dipeptide Isosteres by Means of ?-Lactam Synthon Method -- Synthesis of a Versatile Peptidomimetic Scaffold -- An Asymmetric Synthesis Protocol to Prepare Topographically Constrained ?-Substituted Aromatic Amino Acids -- Synthesis of Oligopeptides Containing an Oxirane Ring in the Place of a Peptidic Bond -- Synthesis of Protected Lactam-Bridged Dipeptides -- Synthesis of Peptidomimics Through Sugar-Based Scaffolds -- The Synthesis of Bicyclic Piperazinone and Related Derivatives -- Synthesis of Dipeptides with ?[CH20] Amide Bond Mimetics -- SNAr-Based Cycloetherification Methodology: Application in the Synthesis of Heterodectic Macrocyclic Peptides with Endo Aryl-Aryl and Aryl-Alkyl Ether Bonds -- Cyclic Aromatic Amino Acids with Constrained ?1 and ?2 Dihedral Angles -- Asymmetric Syntheses of Unnatural Amino Acids and Hydroxyethylene Peptide Isosteres -- Fluoroolefin Isosteres -- Synthesis of 3-Amino-l-CarboxymethyI-Benzodiazepine (BZA) Peptidomimetics -- A Conformationally Restricted ?-Strand HIV Protease Inhibitor -- Synthesis of Cyclopropane-Containing Leu-Enkephalin Analogs -- The 1,5-Disubstituted Tetrazole Ring as a cis-Amide Bond Surrogate -- Synthesis of (2R, 3R, 4R, 5S)-5-tert-Butyloxycarbonylamino-3,4-Dihydroxy-2-1sopropyl-3,4-O,O-Isopropylidene-6-CyctohexyI-Hexanoic Acid -- Synthesis of (2S, 4S, 5S)-5-(t-Butoxycarbonylamino)-4-(t-Butyldimethylsilyloxy)-2-Isopropyl-7-Methyl Octanoic Acid -- Synthesis of ?-Vinyl Amino Acids -- A Novel Synthetic Protocol for the Preparation of Enantiopure 3-, 4-, and 5-Substituted Prolines -- Synthesis of Aminobenzoic Acid-Based Nonpeptide Templates -- Aminimides as Peptidomimetics.
Keywords: Medicinal chemistry; Medicinal Chemistry