Transporters as Targets for Drugs - Napier, Susan; Bingham, Matilda; SpringerLink (Online service) (Berlin, Heidelberg : Springer Berlin Heidelberg : Imprint: Springer, 2009)
Overview: Transporters as Targets for Drug Discovery -- Membrane Transporters: Structure, Function and Targets for Drug Design -- Design of Monoamine Reuptake Inhibitors: SSRIs, SNRIs and NRIs -- Atypical Dopamine Uptake Inhibitors that Provide Clues About Cocaine's Mechanism at the Dopamine Transporter -- The Design, Synthesis and Structure-Activity Relationship of Mixed Serotonin, Norepinephrine and Dopamine Uptake Inhibitors -- Molecular Imaging of Transporters with Positron Emission Tomography -- Pharmacology of Glutamate Transport in the CNS: Substrates and Inhibitors of Excitatory Amino Acid Transporters (EAATs) and the Glutamate/Cystine Exchanger System x c ? -- Glycine Transporters and Their Inhibitors.
Keywords: Human physiology; Pharmacology; Organic chemistry; Medicinal chemistry; Molecular biology; Human Physiology; Pharmacology/Toxicology.; Organic Chemistry; Medicinal Chemistry; Molecular Medicine