Combinatorial Library : Methods and Protocols /

Detalles Bibliográficos
Autor Corporativo: SpringerLink (Online service)
Otros Autores: English, Lisa B. (Editor )
Formato: eBook
Lenguaje:English
Publicado: Totowa, NJ : Humana Press : Imprint: Humana, 2002.
Edición:1st ed. 2002.
Colección:Methods in Molecular Biology, 201
Materias:
Tabla de Contenidos:
  • Library Synthesis and Quality Control
  • Using a Noncovalent Protection Strategy to Enhance Solid-Phase Synthesis
  • Quality Control of Solid-Phase Synthesis by Mass Spectrometry
  • Preparation of Encoded Combinatorial Libraries for Drug Discovery
  • Simple Tools for Manual Parallel Solid Phase Synthesis
  • Cleavage of Compounds from Solid Phase by Gaseous Reagents
  • Synthesis of DNA-Binding Polyamides
  • The Preparation of Phenyl-stilbene Derivatives Using the Safety Catch Linker
  • Host—Guest Chemistry
  • Automated Structure Verification of Small Molecules Libraries Using 1D and 2D NMR Techniques
  • Rapid Liquid-Phase Combinatorial Synthesis of Heterocyclic Libraries
  • Soluble Polymer-Supported Methods for Combinatorial and Organic Synthesis
  • Analytical Methods for Optimization and Quality Control of Combinatorial Synthesis
  • Library Purification and Screening
  • Resolving Racemic Mixtures Using Parallel Combinatorial Libraries
  • Ligand Libraries for the Extraction of Metal Ions
  • Automated Liquid-Liquid Extraction and Ion-Exchange Solid-Phase Extraction for Initial Purification
  • On-Bead and Solution Screening Approaches for Genomically Derived Targets
  • Computational Library Design
  • Design of Virtual Combinatorial Libraries
  • Approaches to Library Design for Combinatorial Chemistry
  • Reagent-Based and Product-Based Computational Strategies in Library Design
  • Designing Combinatorial Libraries for Efficient Screening
  • Application of Neural Networks to Large Dataset QSAR, Virtual Screening, and Library Design.